Creative Biolabs

Aripiprazole [Partial dopamine D2 Agonist]

[CAT#: MOD2005ZP985]

Partial dopamine D2 agonist

Target:
DRD2

Datasheet MSDS Request COA

Certificate of Analysis Lookup
To download a Certificate of Analysis, please enter a lot number in the search box below. Note: Certificate of Analysis not available for kit components.
Lot Number

Bulk Quote
Description
Dopamine D2 partial agonist. Ki (nM) values ​​are 265 (D1), 0.34 (D2), 0.8 (D3), 44 (D4), 1.7 (5-HT1A), 3.4 (5-HT2A), 15 (5-HT2C), 214 (5 -HT6), 39 (5-HT7), 57 (α1), 791 (α2), 61 (H1) and> 1000 (M1). Antipsychotic and antidepressant activity. Central activity after oral administration.
Chemical Name
7-[4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butoxy]-3,4-dihydro-2(1H)-quinolinone
Modulator Type
Agonist
Research Areas
GPCR
Pathways
GPCR Signaling
Molecular Weight
448.39
Chemical Formula
C23H27Cl2N3O2
Source
Synthetic
Solubility
Soluble in DMSO to 100 mM
CAS NO.
129722-12-9
Purity
> 99%
Storage
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months.
Handling Advice
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.

Toxic, refer to SDS for further information.

Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
Target
DRD2
Official Name
DRD2
Full Name
Dopamine receptor D2
Alternative Names
DRD2; D2DR; D2R; dopamine receptor D2
Gene ID
1813(Human); 13489(Mouse); 24318(Rat)
Uniprot ID
P14416(Human); P61168(Mouse); P61169(Rat)
Neural Proteins & Peptides
Neural Antibodies
Neural Cell Lines
Modulators
Biomaterials
Neural Assays
For Research Use Only. Not For Clinical Use.
Send Inquiry Send Inquiry
Inquiry Basket
compare

Go to compare