Creative Biolabs

UNC 0224 [GLP / G9a HMTase Inhibitor]

[CAT#: MOD2005ZP616]

A highly potent, selective G9a HMTase inhibitor

Target:
G9a / GLP HMTases

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Description
An efficient and selective G9a histone lysine methyltransferase (HMTase) inhibitor (IC50 = 15 nM).
Synonyms
Compound 8
Chemical Name
7-[3-(Dimethylamino)propoxy]-2-(hex ahydro-4-methyl-1H-1,4-diazepin-1-yl)-6-methoxy-N- (1-methyl-4-piperidinyl)-4-quinazolinamine
Modulator Type
Inhibitor
Relevant Disease
Neurological Disorders
Molecular Weight
866.19
Chemical Formula
C26H43N7O2
SMILES
CN(CC4)CCC4NC1=C2C(C=C(OCCCN(C)C)C(OC)=C2)=NC(N3CCCN(C)CC3)=N1
Solubility
Soluble in DMSO (100mM)
CAS NO.
1197196-48-7
PubChem Substance ID
44251522
Purity
>98%
Storage
+4°C
Shipping
Room Temperature
Research Use Only
For research use only
Target
G9a / GLP HMTases
Official Name
G9a / GLP HMTases
Alternative Names
G9a / GLP HMTases

For Research Use Only. Not For Clinical Use.
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